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Christoph Lengauer Selected Research

fisogatinib

12/2019First-in-Human Phase I Study of Fisogatinib (BLU-554) Validates Aberrant FGF19 Signaling as a Driver Event in Hepatocellular Carcinoma.
12/2019Acquired On-Target Clinical Resistance Validates FGFR4 as a Driver of Hepatocellular Carcinoma.

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Christoph Lengauer Research Topics

Disease

38Neoplasms (Cancer)
12/2019 - 04/2002
6Colorectal Neoplasms (Colorectal Cancer)
09/2009 - 08/2002
5Carcinogenesis
09/2014 - 01/2008
3Medulloblastoma
09/2010 - 02/2005
2Hepatocellular Carcinoma (Hepatoma)
12/2019 - 04/2015
2Gastrointestinal Stromal Tumors (Gastrointestinal Stromal Tumor)
01/2019 - 11/2017
2Systemic Mastocytosis
01/2019 - 11/2017
2Inborn Genetic Diseases (Disease, Hereditary)
09/2015 - 05/2005
2Multiple Myeloma
02/2011 - 07/2010
2Neoplasm Metastasis (Metastasis)
03/2004 - 11/2003
1Vomiting
12/2019
1Nausea
12/2019
1Disease Progression
12/2019
1Diarrhea
12/2019
1Papillary Thyroid Cancer
01/2018
1Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
01/2018
1medullary Thyroid cancer
01/2018
1Thyroid Neoplasms (Thyroid Cancer)
01/2018
1Melanoma (Melanoma, Malignant)
01/2016
1Carcinosarcoma
09/2014
1Brain Neoplasms (Brain Tumor)
09/2010
1Hypersensitivity (Allergy)
06/2006
1Colonic Neoplasms (Colon Cancer)
11/2004
1Microsatellite Instability
11/2002
1Chromosomal Instability (Chromosome Stability)
11/2002

Drug/Important Bio-Agent (IBA)

11Phosphotransferases (Kinase)IBA
12/2019 - 06/2003
4Protein Isoforms (Isoforms)IBA
01/2016 - 01/2008
4Proteins (Proteins, Gene)FDA Link
09/2015 - 11/2004
4Small Interfering RNA (siRNA)IBA
07/2010 - 07/2007
3avapritinibIBA
01/2019 - 11/2017
3Phosphoric Monoester Hydrolases (Phosphatases)IBA
02/2014 - 11/2003
3DNA (Deoxyribonucleic Acid)IBA
11/2002 - 04/2002
2fisogatinibIBA
12/2019 - 12/2019
2Mitogen-Activated Protein Kinase Kinases (MEKs)IBA
01/2016 - 05/2009
2Messenger RNA (mRNA)IBA
04/2015 - 11/2003
2PyrimidinonesIBA
02/2014 - 05/2012
2TensinsIBA
02/2014 - 05/2012
2Carrier Proteins (Binding Protein)IBA
09/2010 - 11/2004
2Polycomb-Group ProteinsIBA
07/2010 - 02/2009
2Complement System Proteins (Complement)IBA
07/2003 - 07/2003
1midostaurinIBA
01/2019
1Tyrosine Kinase InhibitorsIBA
01/2019
1pralsetinibIBA
01/2018
1Receptor Protein-Tyrosine Kinases (Tyrosine Kinase Receptors)IBA
01/2018
1VemurafenibIBA
01/2016
1MAP Kinase Kinase Kinases (MAP Kinase Kinase Kinase)IBA
01/2016
12- (2- (2- methyl- 2,3- dihydroindol- 1- yl)- 2- oxoethyl)- 6- morpholin- 4- yl- 3H- pyrimidin- 4- oneIBA
01/2016
1AZD 6244IBA
01/2016
1Proto-Oncogene Proteins B-rafIBA
01/2016
1Fibroblast Growth Factors (Fibroblast Growth Factor)IBA
04/2015
1BLU9931IBA
04/2015
1Type 4 Fibroblast Growth Factor ReceptorIBA
04/2015
1ChromatinIBA
09/2014
1RNA (Ribonucleic Acid)IBA
09/2014
1MorpholinosIBA
03/2014
1ThiazolesIBA
03/2014
1AmidesIBA
02/2014
1indolineIBA
02/2014
1BenzoxazolesIBA
05/2012
1benzimidazoleIBA
05/2012
1Transcription Factors (Transcription Factor)IBA
02/2011
1Heterocyclic Compounds (Compounds, Heterocyclic)IBA
02/2011
1Cyclin-Dependent Kinases (cdk Proteins)IBA
02/2011
1Smoothened ReceptorIBA
09/2010
1Heterotrimeric GTP-Binding Proteins (Heterotrimeric G-Proteins)IBA
09/2010
1sonidegibIBA
09/2010
1Guanosine Triphosphate (GTP)IBA
09/2010
1Phosphatidylinositol 3-Kinase (1 Phosphatidylinositol 3 Kinase)IBA
09/2010
1Glucose (Dextrose)FDA LinkGeneric
09/2009
1Cyclin D1IBA
03/2009
1CyclinsIBA
03/2009
1PTEN Phosphohydrolase (PTEN Phosphatase)IBA
09/2008
1LipidsIBA
09/2008
1Phosphatidylinositols (Phosphatidylinositol)IBA
01/2008
13-aminobenzamideIBA
06/2006
1Melphalan (Alkeran)FDA LinkGeneric
06/2006
1Hydrogen Peroxide (Hydroperoxide)FDA LinkGeneric
06/2006
1Etoposide (VP 16)FDA LinkGeneric
06/2006
1GemcitabineFDA Link
06/2006
1Oxaliplatin (Eloxatin)FDA LinkGeneric
06/2006
1NU 1025IBA
06/2006
1Protein Serine-Threonine Kinases (Protein-Serine-Threonine Kinase)IBA
08/2005
1Phosphatidylinositol 3-Kinases (PI 3 Kinase)IBA
08/2005
1CarcinogensIBA
06/2005
12- amino- 1- methyl- 6- phenylimidazo(4,5- b)pyridineIBA
06/2005
1Tretinoin (Retinoic Acid)FDA LinkGeneric
02/2005
1CaspasesIBA
11/2004
1Inhibitor of Apoptosis ProteinsIBA
11/2004
1Non-Steroidal Anti-Inflammatory Agents (NSAIDs)IBA
11/2004
1Fluorouracil (Carac)FDA LinkGeneric
03/2004
1Thymidylate SynthaseIBA
03/2004
1Tyrosine (L-Tyrosine)FDA Link
11/2003
1Calcibiotic Root Canal SealerIBA
11/2003
1EnzymesIBA
04/2002

Therapy/Procedure

13Therapeutics
01/2018 - 02/2005
1Precision Medicine
01/2018
1Immunotherapy
05/2015
1Bone Marrow Transplantation (Transplantation, Bone Marrow)
03/2005
1Chemoprevention
11/2004
1Drug Therapy (Chemotherapy)
03/2004